Amoxicillin Trihydrate (61336-70-7)
Bayani
● Amoxicillin Trihydrate (61336-70-7)
● CAS No.: 61336-70-7
● EINECS Lamba: 248-003-8
● MF: C16H19N3O5S
● Kunshin: 25kg/drum
Cikakken Bayani
Amoxicillin trihydrate, penicillin mai faɗaɗaɗaɗaɗɗen roba, yana da bakan ƙwayoyin cuta iri ɗaya, tasiri da aikace-aikace kamar ampicillin.Amoxicillin trihydrate shine hydrate wanda shine nau'in trihydrate na amoxicillin;maganin rigakafi na semisynthetic, wanda aka yi amfani da shi kadai ko a hade tare da potassium clavulanate (a karkashin sunan kasuwanci Augmentin) don maganin cututtuka iri-iri.Yana da matsayi a matsayin maganin ƙwayar cuta da kuma wakili na antimicrobial.Ya ƙunshi amoxicillin.Amoxicillin wani nau'i ne mai faɗin bakan, maganin rigakafi na aminopenicillin semisynthetic tare da ayyukan ƙwayoyin cuta.Amoxicillin yana ɗaure kuma yana hana furotin mai ɗaure penicillin (PBP) 1A wanda ke kan membrane na ciki na bangon ƙwayoyin cuta.Rashin kunnawa na PBPs yana tsoma baki tare da haɗin giciye na sarƙoƙi na peptidoglycan waɗanda suka wajaba don ƙarfin bangon ƙwayoyin ƙwayoyin cuta da rigidity.Wannan yana katse haɗin bangon ƙwayoyin ƙwayoyin cuta kuma yana haifar da rauni na bangon ƙwayoyin ƙwayoyin cuta kuma yana haifar da tantanin halitta.
An gano Amoxicillin a cikin 1958 kuma ya fara amfani da magani a cikin 1972. An amince da Amoxil don amfani da magani a Amurka a 1974, kuma a cikin Burtaniya a 1977. Yana cikin Jerin Mahimman Magunguna na Hukumar Lafiya ta Duniya (WHO). yana daya daga cikin magungunan kashe kwayoyin cuta da aka fi rubutawa ga yara.Ana samun Amoxicillin azaman magani na gama-gari. A cikin 2020, shine magani na 40 da aka fi ba da izini a Amurka, tare da rubutattun magunguna sama da miliyan 15.
Aikace-aikace
Ana amfani da shi don magance cututtukan ƙwayoyin cuta, kamar cututtukan ƙirji (ciki har da ciwon huhu) da ƙurar haƙora.Hakanan ana iya amfani dashi tare da sauran maganin rigakafi da magunguna don magance ciwon ciki.Sau da yawa ana wajabta wa yara, don magance ciwon kunne da ciwon kirji.
Sharuɗɗan gwaji | Matsayi | Sakamako |
Assay | 95.0% ~ 102.0% | 99.9% |
PH | 3.5 ~ 5.5 | 4.6 |
Bayyanar mafita | 0.5mol/L HCL≤2# 2mol/L NH4 OH≤2# | 1#1# |
Ruwa | 11.5% ~ 14.5% | 13.2% |
Abubuwan da ke da alaƙa | Rashin tsarki (max.)≤1.0% | 0.13% |
Takamaiman jujjuyawar gani | +290''~+315'' | +305° |
Sulfated ash | ≤1.0% | 0.1% |
NN-Dimethylannline | ≤20ppm | Ba a taɓa amfani da shi wajen samarwa ba |
Methylen chloride | ≤600ppm | 296pm |
Triethylamine | ≤320ppm | 155pm |
Acetone | ≤3000ppm | 95ppm ku |
Ƙarshe: Ya dace da Matsayin EP 6th. |